transformation of 2-benzoylamino-1-(?-naphthyl)propan-1-ol into 4-methyl-1-phenyl benzo[f] isoquinoline rather than its 3-substituted isomer
نویسندگان
چکیده
the necessary conditions to transform hydroxyamide (1) and 2-oxazolines (2, 3) into 3- or 4-methyl benzo[f] isoquinolines (4, 5) has been established. the mechanism of these reactions has been proposed claiming the existence of the protonated 2-oxazoline (6) and the styrylamides (7) as intermediates.
منابع مشابه
TRANSFORMATION OF 2-BENZOYLAMINO-1-(?-NAPHTHYL)PROPAN-1-OL INTO 4-METHYL-1-PHENYL BENZO[f] ISOQUINOLINE RATHER THAN ITS 3-SUBSTITUTED ISOMER
The necessary conditions to transform hydroxyamide (1) and 2-oxazolines (2, 3) into 3- or 4-methyl benzo[f] isoquinolines (4, 5) has been established. The mechanism of these reactions has been proposed claiming the existence of the protonated 2-oxazoline (6) and the styrylamides (7) as intermediates.
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عنوان ژورنال:
journal of sciences islamic republic of iranجلد ۱۲، شماره ۱، صفحات ۰-۰
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